Preliminary Screening for Anti-Inflammatory, Anti-Nociceptive and Antioxidant Activities of Five New Synthesized Paratoluene Sulphonamide Derivatives of Amino Acids
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[1] R. Davicino et al., Different activities of Schinus areira L.: anti-inflammatory or pro-inflammatory effect, Immunopharmacol. Immunotoxicol. 32(4) (2010) 620-627.
[2] A. N, Shikov et al., Anti-inflammatory effect of Pinus sibirica oil extract in animal models, J. Nat. Med. 62 (2008) 436–440.
[3] S. Ahmad et al., Synthesis and biological evaluation of some novel 6-aryl-2-(p-sulfamylphenyl)-4, 5-dihydropyridazin-3(2H)-ones as anti-cancer, antimicrobial, and anti-inflammatory agents, J. Enzyme Inhib. Med. Chem. 25 (2010) 266–271.
[4] A.G. Habeeb, P.N. Praveen Rao, E.E. Knaus, Design and Synthesis of Celecoxib and Rofecoxib Analogues as Selective Cyclooxygenase-2 (COX-2) Inhibitors: Replacement of Sulfonamide and Methylsulfonyl Pharmacophores by an Azido Bioisostere, J. Med. Chem. 44 (2001).
[5] A. Casini, A. Scozzafava, C.T. Supuran, Sulfonamide derivatives with protease inhibitory action as anticancer, anti-inflammatory and antiviral agents, Exp. Opin. Ther. Pat. 12 (2002) 1307-1327.
DOI: https://doi.org/10.1517/13543776.12.9.1307[6] A. Kołaczek et al., Biological activity and synthesis of sulfonamide derivatives: a brief review, Chemik. 68 (2014) 620–628.
[7] N. Anand, Sulfonamides and Sulfons, In M.E. Wolff (Ed. ), Burger's Medicinal Chemistry, Vol. 2, 5th ed, New York, Wiley- Interscience, 1996, Chapter 33.
[8] C.B.C. Ikpa, U.C. Okoro, Synthesis of new paratoluene sulphonamide derivatives of amino acids and their anti bacterial activities, IOSR Journal of Applied Chemistry. 9 (6) (Ver. II) (2016) 31-34.
[9] J.W. Ward, J.R. Elsea, Animal case and use in drug fate and metabolism, In: R.G. Edward, L.H. Jean, (Eds), Methods and Techniques, 1st edi. New York, Markel Dekker, (1997).
[10] Organization for Economic Cooperation and Development, OECD guidelines for the testing of chemicals, acute oral toxicity - up-and down procedure, No. 425. Paris, Organization for Economic Cooperation and Development, 2008. [Online] Available from: http: /www. oecd-ilibrary. org/docserver/download/9742501e. pdf?expires=1437730561&id=id&accname=guest&checksum=0B6C86B8F1B2E751997E5F54CFDF8F5E [Accessed on 5th May, 2015].
[11] B. Adzu et al., Anti-inflammatory and antinociceptive effects of Sphaeranthus senegalensis, J. Ethnopharmacol. 84 (2003) 169–173.
[12] M.A. Alam et al., Antinociceptive and anti-inflammatory properties of Ruellia tuberosa, Pharm. Biol. 47 (3) (2009) 209-214.
[13] M.I. Ezeja et al., Anti-inflammatory and Antioxidant Activities of the Methanolic Leaf Extract of Cissus aralioides, Am. J. Pharmacol. Sci. 3 (2015) 1-6.
[14] F.F. Benzie, J.J. Strain, Ferric reducing/Antioxidant power Assay: Direct measure of total antioxidant activity of biological fluids and modified version for simultaneous measurement of total antioxidant power and ascorbic acid concentration, Methods Enzymol. 299 (1999).
[15] S.O. Onoja et al., Antioxidant, anti-inflammatory and antinociceptive activities of methanolic extract of Justicia secunda Vahl leaf, Alex. J. Med. (2016) in press. http: /dx. doi. org/10. 1016/j. ajme. 2016. 06. 001.
[16] F. C Vilela et al., Anti-inflammatory and antipyretic effects of Sonchus oleraceus in rats, J. Ethnopharmacol. 127 (2010) 737–741.
[17] I.C. Obidike et al., The anti-inflammatory and antinociceptive properties of the chloroform fraction from Phyllanthus niruri plant is mediated via the peripheral nervous system, J. Diet. Suppl. 7 (4) (2010) 341-350.
[18] M.S. Brandão et al., Antinociceptive effect of lecythis pisonis camb. (lecythidaceae) in models of acute pain in mice, J. Ethnopharmacol. 146 (2013) 180-186.
[19] A.O.T. Ashafa et al., Evaluation of aqueous extract of Felicia muricata leaves for anti-inflammatory, antinociceptive, and antipyretic activities, Pharm. Biol. 48(9) (2010) 994-1001.